Vilanterol trifenatate
Cat. No.:YN320847
CAS No. :503070-58-4
产品名称: | Vilanterol trifenatate |
CAS No.: | 503070-58-4 |
Chemical Name: | Benzeneacetic acid, α,α-diphenyl-, compd. with (α1R)-α1-[[[6-[2-[(2,6-dichlorophenyl)methoxy]ethoxy]hexyl]amino]methyl]-4-hydroxy-1,3-benzenedimethanol; |
Synonyms: | GW642444 trifenatate |
分子量: | 774.77 |
分子式: | C₄₄H₄₉Cl₂NO₇ |
SMILES: | OC1=CC=C([C@@H](O)CNCCCCCCOCCOCC2=C(Cl)C=CC=C2Cl)C=C1CO.O=C(O)C(C3=CC=CC=C3)(C4=CC=CC=C4)C5=CC=CC=C5 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Vilanterol trifenatate (GW642444 trifenatate) 是一种长效的β2-AR激动剂,效力持续24小时。 对β2-AR,β1-AR和β3-AR的pEC50分别为10.37,6.98 ,7.36。 |
IC50和靶点: | |
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Procopiou, P., et al.: J. Med. Chem., 53, 4522 (2010)
Kempsford, R., et al.: Pulm. Pharmacol. Ther., 26, 256 (2013)