Cabamiquine succinate
Cat. No.:YN252299
| 产品名称: | Cabamiquine succinate |
| CAS No.: | 2444781-71-7 |
| Chemical Name: | |
| Synonyms: | DDD107498 succinate; DDD-498 succinate; M5717 succinate |
| 分子量: | 580.65 |
| 分子式: | C31H37FN4O6 |
| SMILES: | 暂无 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Cabamiquine (DDD107498) succinate 是一种有效、可口服的抗疟疾 (antimalarial) 剂,能够抑制寄生虫生命周期的多个阶段,对P. falciparum3D7 的EC50值为 1 nM。Cabamiquine succinate 通过靶作用于eEF2/CaMKIII来抑制蛋白合成,对 WT-PfeEF2 的EC50值为 2 nM。 |
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