Entinostat
Cat. No.：YN270147
CAS No. ：209783-80-2
| 产品名称: | Entinostat |
| CAS No.: | 209783-80-2 |
| Chemical Name: | N-[[4-[[(2-aminophenyl)amino]carbonyl]phenyl]methyl]-carbamic acid, 3-pyridinylmethyl ester |
| Synonyms: | 恩替诺特; MS-275; SNDX-275 |
| 分子量: | 376.41 |
| 分子式: | C₂₁H₂₀N₄O₃ |
| SMILES: | O=C(NCC1=CC=C(C=C1)C(NC2=CC=CC=C2N)=O)OCC3=CC=CN=C3 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Entinostat 选择性，可口服的HDAC class I抑制剂，抑制HDAC1，HDAC2和HDAC3的IC50分别为 243 nM，453 nM 和 248 nM。 |
| IC50和靶点: | [{name:"HDAC1:243 nM (IC50)"},{name: "HDAC3:248 nM (IC50)"},{name: "HDAC2:453 nM (IC50)"}] |
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