PR-39
Cat. No.:YN251824
产品名称: | PR-39 |
CAS No.: | 139637-11-9 |
Chemical Name: | |
Synonyms: | RRRPRPPYLPRPRPPPFFPPRLPPRIPPGFPPRFPPRFP-NH2 |
分子量: | 4719.74 |
分子式: | C₂₂₉H₃₄₆N₇₀O₄₀ |
SMILES: | 暂无 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | PR-39 是富含脯氨酸和精氨酸的天然抗菌肽,是一种非竞争性,可逆和变构的蛋白酶体 (proteasome) 抑制剂。PR-39 可逆地结合到蛋白酶体的 α7 亚基上,并通过泛素-蛋白酶体途径阻断 NF-κB 抑制剂 IκBα 的降解。PR-39 刺激小鼠的血管生成,抑制炎症反应并显着减小心肌梗死面积。 |
IC50和靶点: | |
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