JWG-071
Cat. No.:YN350060
| 产品名称: | JWG-071 |
| CAS No.: | 2250323-50-1 |
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| 分子量: | 612.76 |
| 分子式: | C₃₄H₄₄N₈O₃ |
| SMILES: | COC1=CC(C(N2CCC(N3CCN(C)CC3)CC2)=O)=CC=C1NC4=NC=C(N(C)C5=O)C(N(C6=CC=CC=C65)C(C)CC)=N4 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | JWG-071 是首次报道的ERK5激酶选择性化学探针。JWG-071 提高了 ERK5 活性和 BRD4 选择性。JWG-071 将是反卷积 ERK5 和 BRD4 药理学急需的化学探针。 |
| IC50和靶点: | [{name:"ERK5:88 nM (IC50)"}] |
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