Fz7-21
Cat. No.:YN450204
产品名称: | Fz7-21 |
CAS No.: | 2247635-23-8 |
Chemical Name: | |
Synonyms: | Ac-LPSDDLEFWCHVMY-NH2 |
分子量: | 1796.05 |
分子式: | C83H114N18O23S2 |
SMILES: | 暂无 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Fz7-21 (Ac-LPSDDLEFWCHVMY-NH2) 是一种有效的FZD7受体的肽拮抗剂,选择性地结合到 FZD7 CRD 亚类,并改变 CRD 的构象及其脂质结合槽的结构。人和小鼠 FZD7 CRD 的EC50值分别为 58 和 34 nM。Fz7-21 损害 FZD7 在 Wnt-β-catenin 信号传导中的功能和肠类器官中的干细胞功能。 |
IC50和靶点: | |
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Clinical Trial: | |
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