HTH-01-091
Cat. No.:YN270691
| 产品名称: | HTH-01-091 | 
| CAS No.: | 2000209-42-5 | 
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| 分子量: | 499.43 | 
| 分子式: | C26H28Cl2N4O2 | 
| SMILES: | 暂无 | 
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. | 
| 运输: | Room temperature in continental US; may vary elsewhere. | 
| 产品描述: | HTH-01-091 是一种强效且选择性的maternal embryonic leucine zipper kinase (MELK)抑制剂,其IC50为 10.5 nM。HTH-01-091 还能抑制PIM1/2/3、RIPK2、DYRK3、smMLCK和CLK2。HTH-01-091 可用于乳腺癌研究。 | 
| IC50和靶点: | [{name:"DYRK4:41.8 nM (IC50)"},{name: "PIM1:60.6 nM (IC50)"},{name: "mTOR:632 nM (IC50)"},{name: "CDK7:1230 nM (IC50)'}, 'PIM2', 'PIM3'] | 
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