GSK-872 hydrochloride
Cat. No.:YN270727
CAS No. :2703752-81-0
产品名称: | GSK-872 hydrochloride |
CAS No.: | 2703752-81-0 |
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分子量: | 419.94 |
分子式: | C19H18ClN3O2S2 |
SMILES: | 暂无 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | GSK-872 hydrochloride 是RIPK3抑制剂,高亲和力结合 RIP3 激酶结构域,IC50为1.8 nM,并抑制激酶活性,IC50为1.3 nM。GSK-872 hydrochloride 降低RIPK3介导的坏死 (necroptosis) 和随后的 HMGB1 的细胞质易位和表达,并改善早期脑损伤中的脑水肿和神经功能缺损。 |
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