TNIK-IN-3
Cat. No.:YN270728
CAS No. :2754265-25-1
产品名称: | TNIK-IN-3 |
CAS No.: | 2754265-25-1 |
Chemical Name: | |
Synonyms: | |
分子量: | 387.41 |
分子式: | C23H18FN3O2 |
SMILES: | 暂无 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | TNIK-IN-3 (化合物 21k) 是一种有效,选择性和具有口服活性的TNIK抑制剂,IC50值为 0.026 μM。TNIK-IN-3 还可以抑制Flt4(IC50=0.030 μM),Flt1(IC50=0.191 μM) 和DRAK1(IC50=0.411 μM)。TNIK-IN-3 可用于结直肠癌的研究。 |
IC50和靶点: | |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |