Famitinib
Cat. No.:YN270796
| 产品名称: | Famitinib | 
| CAS No.: | 1044040-56-3 | 
| Chemical Name: | |
| Synonyms: | 法米替尼; SHR1020 | 
| 分子量: | 暂无 | 
| 分子式: | 暂无 | 
| SMILES: | 暂无 | 
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. | 
| 运输: | Room temperature in continental US; may vary elsewhere. | 
| 产品描述: | Famitinib (SHR1020) 是一种有效的,具有口服活性的多靶点激酶抑制剂,抑制c-kit,VEGFR-2和PDGFRβ的活性,IC50值分别为 2.3 nM、4.7 nM 和 6.6 nM。Famitinib具有抗肿瘤活性。且诱导细胞凋亡 (apoptosis)。 | 
| IC50和靶点: | [{name:"VEGFR-2:4.2 nM (IC50)"},{name: "PDGFRβ:6.6 nM (IC50)"},{name: "c-kit:2.3 nM (IC50)"}] | 
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |