Aspidin BB
Cat. No.:YN270818
| 产品名称: | Aspidin BB | 
| CAS No.: | 2361988-77-2 | 
| Chemical Name: | |
| Synonyms: | |
| 分子量: | 暂无 | 
| 分子式: | 暂无 | 
| SMILES: | 暂无 | 
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. | 
| 运输: | Room temperature in continental US; may vary elsewhere. | 
| 产品描述: | cRIPGBM chloride 是一种口服有效的促凋亡衍生物,cRIPGBM 可从多形性胶质母细胞瘤 (GBM) 癌症干细胞 (CSC) 中产生。cRIPGBM chloride 靶向受体相互作用蛋白激酶 2 (RIPK2) 以诱导半胱天冬酶caspase 1依赖性细胞凋亡。cRIPGBM chloride 抑制RIPK2/TAK1(促存活复合物) 的形成,并增加RIPK2/caspase 1(促凋亡复合物) 的形成。cRIPGBM chloride 在动物模型中发挥了强力的体内抗肿瘤活性。 | 
| IC50和靶点: | |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |