Thioperamide
Cat. No.:YN320563
产品名称: | Thioperamide |
CAS No.: | 106243-16-7 |
Chemical Name: | |
Synonyms: | MR-12842 |
分子量: | 292.44 |
分子式: | C₁₅H₂₄N₄S |
SMILES: | S=C(N1CCC(C2=CN=CN2)CC1)NC3CCCCC3 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Thioperamide (MR-12842) 是一种有效的,具有口服活性的,可透过血脑屏障的选择性H3受体拮抗剂,抑制 [3H] 组胺释放的Ki为 4.3 nM。Thioperamide 抑制 [3H] 组胺合成的Ki为 31 nM 。 |
IC50和靶点: | |
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