Bilastine
Cat. No.:YN320871
CAS No. :202189-78-4
产品名称: | Bilastine |
CAS No.: | 202189-78-4 |
Chemical Name: | 4-[2-[4-[1-(2-ethoxyethyl)-1H-benzimidazol-2-yl]-1-piperidinyl]ethyl]-α,α-dimethyl-benzeneacetic acid |
Synonyms: | 比拉斯汀 |
分子量: | 463.61 |
分子式: | C₂₈H₃₇N₃O₃ |
SMILES: | CC(C)(C1=CC=C(CCN2CCC(C3=NC4=CC=CC=C4N3CCOCC)CC2)C=C1)C(O)=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Bilastine是组胺H1受体拮抗剂,可作用于变应性鼻结膜炎和荨麻疹。 |
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Corcóstegui, R., Labeaga, L., Innerárity, A., et al.Preclinical pharmacology of bilastine, a new selective histamine H1 receptor antagonist: Receptor selectivity and in vitro antihistaminic activityDrugs R. D.6(6),371-384(2005)
Corcóstegui, R., Labeaga, L., Innerárity, A., et al.In vivo pharmacological characterisation of bilastine, a potent and selective histamine H1 receptor antagonistDrugs R. D.7(4),219-231(2006)