BRD9757
Cat. No.:YN290628
| 产品名称: | BRD9757 |
| CAS No.: | 1423058-85-8 |
| Chemical Name: | |
| Synonyms: | BRD 9757 |
| 分子量: | 127.143 |
| 分子式: | C6H9NO2 |
| SMILES: | 暂无 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | BRD9757 是一种有效的、无帽的、选择性的HDAC6抑制剂,IC50为 30 nM。与 I 类(>20 倍)和 II 类(>400 倍)HDAC 相比,BRD9757 对HDAC6表现出出色的选择性。 |
| IC50和靶点: | [{name:"HDAC6:0.03 μM (IC50)"},{name: "HDAC1:0.638 μM (IC50)"},{name: "HDAC2:1.79 μM (IC50)"},{name: "HDAC3:0.694 μM (IC50)"},{name: "HDAC4:21.80 μM (IC50)"},{name: "HDAC5:18.32 μM (IC50)"},{name: "HDAC7:12.61 μM (IC50)"},{name: "HDAC8:1.09 μM (IC50)"},{name: "HDAC9:>33.33 μM (IC50)"}] |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |