Perospirone
Cat. No.：YN321568
CAS No. ：150915-41-6
规格
价格(RMB)
库存
| 产品名称: | Perospirone |
| CAS No.: | 150915-41-6 |
| Chemical Name: | |
| Synonyms: | 哌罗匹隆; SM-9018 free base |
| 分子量: | 426.57 |
| 分子式: | C₂₃H₃₀N₄O₂S |
| SMILES: | O=C([C@@]1([H])[C@]2([H])CCCC1)N(C2=O)CCCCN3CCN(C4=NSC5=C4C=CC=C5)CC3 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Perospirone (SM-9018 free base) 是具有口服活性的5-HT2A受体 (Ki=0.6 nM) 和多巴胺 D2受体 (Ki=1.4 nM) 的拮抗剂，也是5-HT1A受体 (Ki=2.9 nM) 的部分激动剂。Perospirone 是一种非典型的抗精神病剂，可用于精神分裂症的研究。 |
| IC50和靶点: | [{name:"5-HT2A Receptor:0.6 nM (Ki)"},{name: "Dopamine D2:1.4 nM (Ki)"},{name: "5-HT1A Receptor:2.9 nM (Ki)"},{name: "5-HT1 Receptor:18 nM (Ki)"},{name: "Dopamine D1:41 nM (Ki)"}] |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
