Camonsertib
Cat. No.:YN290722
| 产品名称: | Camonsertib |
| CAS No.: | 2417489-10-0 |
| Chemical Name: | |
| Synonyms: | RP-3500; ATR inhibitor 4 |
| 分子量: | 410.47 |
| 分子式: | C21H26N6O3 |
| SMILES: | 暂无 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Camonsertib (RP-3500) 是一种口服有效的,选择性ATR激酶抑制剂 (ATRi),在生化试验中的IC50为 1.00 nM。Camonsertib 对ATR的选择性是mTOR的 30 倍 (IC50=120 nM),是 ATM、DNA-PK 和PI3Kα激酶的 > 2,000 倍。Camonsertib 具有有效的抗肿瘤活性。 |
| IC50和靶点: | |
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| Solvent & Solubility: |