G-1
Cat. No.：YN480308
CAS No. ：881639-98-1
规格
价格(RMB)
库存
| 产品名称: | G-1 |
| CAS No.: | 881639-98-1 |
| Chemical Name: | rel-1-[4-(6-bromo-1,3-benzodioxol-5-yl)-3aR,4S,5,9bS-tetrahydro-3H-cyclopenta[c]quinolin-8-yl]-ethanone |
| Synonyms: | G 1;G-1 |
| 分子量: | 412.28 |
| 分子式: | C₂₁H₁₈BrNO₃ |
| SMILES: | BrC1=C([C@H]2[C@]3([H])[C@](C=CC3)([H])C4=CC(C(C)=O)=CC=C4N2)C=C5C(OCO5)=C1 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | G-1 是一个非甾体，高亲和力且有选择性的GPR30激动剂，其Ki值为 11 nM。 |
| IC50和靶点: | |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
Revankar, C.M., Cimino, D.F., Sklar, L.A., et al.A transmembrane intracellular estrogen receptor mediates rapid cell signalingScience307,1625-1630(2005)
Bologa, C.G., Revankar, C.M., Young, S.M., et al.Virtual and biomolecular screening converge on a selective agonist for GPR30Nat. Chem. Biol.2(4),207-212(2006)
