Raloxifene 6-Monomethyl Ether
Cat. No.:YN481232
| 产品名称: | Raloxifene 6-Monomethyl Ether | 
| CAS No.: | 178451-13-3 | 
| Chemical Name: | [2-(4-Hydroxyphenyl)-6-methoxybenzo[b]thien-3-yl][4-[2-(1-piperidinyl)ethoxy]phenyl]methanone; | 
| Synonyms: | |
| 分子量: | 487.61 | 
| 分子式: | C₂₉H₂₉NO₄S | 
| SMILES: | O=C(C1=C(C2=CC=C(O)C=C2)SC3=CC(OC)=CC=C31)C4=CC=C(OCCN5CCCCC5)C=C4 | 
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. | 
| 运输: | Room temperature in continental US; may vary elsewhere. | 
| 产品描述: | Raloxifene 6-Monomethyl Ether 是一种 Raloxifene 衍生物,其抑制雌激素受体 α (estrogen receptor α)。Raloxifene 4-Monomethyl Ether 抑制 MCF-7 细胞,IC50为 250 nM,pIC50为 6.6。 | 
| IC50和靶点: | |
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| Solvent & Solubility: | 
Jone, C.D., et al.: J. Med. Chem., 27, 1057 (1984), Buelke-Sam, J., et al.: Reprod. Toxicol., 12, 217 (1998),