Irsogladine maleate
Cat. No.：YN321453
| 产品名称: | Irsogladine maleate |
| CAS No.: | 84504-69-8 |
| Chemical Name: | 6-(2,5-dichlorophenyl)-1,3,5-triazine-2,4-diamine, 2Z-butenedioate |
| Synonyms: | 马来酸伊索拉定; Dicloguamine maleate; MN1695 |
| 分子量: | 372.16 |
| 分子式: | C₁₃H₁₁Cl₂N₅O₄ |
| SMILES: | O=C(O)/C=C\C(O)=O.NC1=NC(N)=NC(C2=CC(Cl)=CC=C2Cl)=N1 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Irsogladine马来酸盐是PDE4抑制剂和毒蕈碱乙酰胆碱受体结合剂。 |
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Kyoi, T., Oka, M., Noda, K., et al.Irsogladine prevents monochloramine-induced gastric mucosal lesions by improving the decrease in mucosal blood flow due to the disturbance of nitric oxide synthesis in ratsJ. Pharmacol. Sci.93(3),314-320(2003)
Ueda, F., Ban, K., and Ishima, T.Irsogladine activates gap-junctional intercellular communication through M1 muscarinic acetylcholine receptorJ. Pharm. Exp. Ther.274(2),815-819(1995)
Kyoi, T., Noda, K., Oka, M., et al.Irsogladine, an anti-ulcer drug, suppresses superoxide production by inhibiting phosphodiesterase type 4 in human neutrophilsLife Sci.76(1),71-83(2004)
