NRA-0160
Cat. No.：YN320169
CAS No. ：204718-47-8
规格
价格(RMB)
库存
| 产品名称: | NRA-0160 |
| CAS No.: | 204718-47-8 |
| Chemical Name: | |
| Synonyms: | |
| 分子量: | 439.52 |
| 分子式: | C₂₄H₂₃F₂N₃OS |
| SMILES: | O=C(C1=NC(C2=CC=C(F)C=C2)=C(CCN3CC/C(CC3)=C\C4=CC=CC(F)=C4)S1)N |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | NRA-0160 是一种选择性的dopamine D4 receptor拮抗剂，Ki值为 0.48 nM；同时对dopamine D2 receptor，D3 receptor，大鼠5-HT2A receptor和α1 adrenoceptor分别具有不同程度的亲和度，Ki值分别为 >10000 nM，39 nM，180 nM 和 237 nM。 |
| IC50和靶点: | [{name:"D4 Receptor:0.48 nM (Ki)"},{name: "D3 Receptor:39 nM (Ki)"},{name: "5-HT2A Receptor:180 nM (Ki, in rat)"},{name: "Rat α1 adrenoceptor:237 nM (Ki)"}] |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
