Ketanserin
Cat. No.：YN320289
CAS No. ：74050-98-9
| 产品名称: | Ketanserin |
| CAS No.: | 74050-98-9 |
| Chemical Name: | 3-[2-[4-(4-fluorobenzoyl)-1-piperidinyl]ethyl]-2,4(1H,3H)-quinazolinedione |
| Synonyms: | 酮色林; R41468 |
| 分子量: | 395.43 |
| 分子式: | C₂₂H₂₂FN₃O₃ |
| SMILES: | O=C(C1=CC=CC=C1N2)N(CCN3CCC(C(C4=CC=C(F)C=C4)=O)CC3)C2=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Ketanserin 是一种选择性的5-HT2 receptor拮抗剂。Ketanserin 也抑制 hERG 电流 (IhERG)，IC50为 0.11 μM，这种作用具有浓度依赖性。 |
| IC50和靶点: | |
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| Solvent & Solubility: |
Leysen, J.E., Awouters, F., Kennis, L., et al.Receptor binding profile of R 41 468, a novel antagonist at 5-HT2 receptorsLife Sci.28(9),1015-1022(1981)
