Risperidone mesylate
Cat. No.:YN320413
| 产品名称: | Risperidone mesylate |
| CAS No.: | 666179-96-0 |
| Chemical Name: | |
| Synonyms: | R 64 766 mesylate |
| 分子量: | 506.59 |
| 分子式: | C₂₄H₃₁FN₄O₅S |
| SMILES: | CS(=O)(O)=O.FC1=CC(ON=C2C3CCN(CCC(C(N(CCCC4)C4=N5)=O)=C5C)CC3)=C2C=C1 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Risperidone mesylate(R 64 766 mesylate) 是5-HT2受体的阻断剂,P-糖蛋白(P-Glycoprotein)的抑制剂 和dopamine D2受体的拮抗剂,其对 5-HT2A和 dopamine D2受体的Ki值分别为 4.8,5.9 nM。 |
| IC50和靶点: | [{name:"5-HT2A Receptor:4.8 nM (Ki)"},{name: "D2 Receptor:5.9 nM (Ki)'}, 'P-glycoprotein'] |
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| Clinical Trial: | |
| Solvent & Solubility: |