GR 125743
Cat. No.:YN320549
CAS No. :148547-33-5
产品名称: | GR 125743 |
CAS No.: | 148547-33-5 |
Chemical Name: | |
Synonyms: | |
分子量: | 416.52 |
分子式: | C₂₅H₂₈N₄O₂ |
SMILES: | O=C(C1=CC=C(C(C)=C1)C2=CC=NC=C2)NC3=CC=C(C(N4CCN(CC4)C)=C3)OC |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | GR 125743 是一种选择性的5-HT1B/1D受体拮抗剂,对 h5-HT1B作用的Kd值为 0.61 nM。GR 125743 可用于帕金森病和心血管疾病的研究。 |
IC50和靶点: | [{name:"human 5-HT1B Receptor:8.85 (pKi)"},{name: "human 5-HT1D Receptor:8.31 (pKi)"}] |
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Clinical Trial: | |
Solvent & Solubility: |