ML 10302 hydrochloride
Cat. No.:YN320870
产品名称: | ML 10302 hydrochloride |
CAS No.: | 186826-17-5 |
Chemical Name: | |
Synonyms: | |
分子量: | 349.25 |
分子式: | C₁₅H₂₂Cl₂N₂O₃ |
SMILES: | O=C(OCCN1CCCCC1)C2=CC(Cl)=C(N)C=C2OC.[H]Cl |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | ML 10302 hydrochloride 是一种高效、选择性的 5-HT4受体 (5-HT4receptor) 激动剂,其EC50值为 4 nM。对 5-HT4的绑定作用比5-HT3强至少 680 倍。 |
IC50和靶点: | [{name:"5-HT4 Receptor:4 nM (EC50)"},{name: "5-HT4 Receptor:1.07 nM (Ki)"},{name: "5-HT3 Receptor:782 nM (Ki)"}] |
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