CYM51010
Cat. No.:YN322141
产品名称: | CYM51010 |
CAS No.: | 1069498-96-9 |
Chemical Name: | 1-[[4-(acetylamino)phenyl]methyl]-4-(2-phenylethyl)-4-piperidinecarboxylic acid, ethyl ester |
Synonyms: | |
分子量: | 408.5 |
分子式: | C25H32N2O3 |
SMILES: | CC(NC(C=C1)=CC=C1CN2CCC(C(OCC)=O)(CCC3=CC=CC=C3)CC2)=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | CYM51010 是 μ 阿片受体-δ 阿片受体异二聚体的一种偏倚配体。CYM51010 可表现出与吗啡相似的抗伤害感受活性,但其耐受性发展和戒断症状的水平有所降低。 |
IC50和靶点: | |
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Pinello, C., Guerrero, M., Eberhart, C., et al.Characterization of an agonist probe for opioid receptor mu 1 (OPRM1)-opioid receptor delta 1 (OPRD1) heterodimerizationProbe Reports from the NIH Molecular Libraries Program,1-14(2012)