CAY10590
Cat. No.：YN322152
| 产品名称: | CAY10590 |
| CAS No.: | 1101136-50-8 |
| Chemical Name: | 4-[(1-oxo-7-phenylheptyl)amino]-(4R)-octanoic acid |
| Synonyms: | GK115 |
| 分子量: | 347.5 |
| 分子式: | C21H33NO3 |
| SMILES: | O=C(N[C@H](CCCC)CCC(O)=O)CCCCCCC1=CC=CC=C1 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | CAY10590 (GK115) 是一种分泌型磷脂酶 A2(sPLA2) 的抑制剂，可用于慢性炎症性肾脏疾病的研究。 |
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Balestrieri, B., and Arm, J.P.Group V sPLA2: Classical and novel functionsBiochim. Biophys. Acta1761,1280-1288(2006)
Antonopoulou, G., Barbayianni, E., Magrioti, V., et al.Structure-activity relationships of natural and non-natural amino acid-based amide and 2-oxoamide inhibitors of human phospholipase A2 enzymesBioorg. Med. Chem.16,10257-10269(2008)
