Dexmedetomidine
Cat. No.：YN322162
| 产品名称: | Dexmedetomidine |
| CAS No.: | 113775-47-6 |
| Chemical Name: | 5-[(1S)-1-(2,3-Dimethylphenyl)ethyl]-1H-imidazole; (S)-4-[1-(2,3-Dimethylphenyl)ethyl]-1H-imidazole; (+)-Medetomidine; (S)-Medetomidine; MPV 1440; d-Medetomidine; |
| Synonyms: | 右美托咪定; (+ |
| 分子量: | 200.28 |
| 分子式: | C13H16N2 |
| SMILES: | 暂无 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Dexmedetomidine ((+)-Medetomidine) 是一种有效，选择性和具有口服活性的 α2 肾上腺素能受体 (α2-adrenoceptor) 激动剂，Ki值为 1.08 nM。Dexmedetomidine 对 α1 肾上腺素受体显示出 1620 倍的选择性。Dexmedetomidine 具有抗焦虑作用，可用于促进睡眠和缓解疼痛的研究。 |
| IC50和靶点: | [{name:"α2-adrenergic receptor:1.08 nM (Ki)"}] |
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| Clinical Trial: | |
| Solvent & Solubility: |
Rajala, R., et al.: Eur. J. Pharm. Sci., 1, 219 (1994), Jalonen, J., et al.: Anesthesiology, 86, 331 (1997), Talke, P., et al.: Anesth. Analg., 85, 1136 (1997), Bhana, N., et al.: Drugs, 59, 263 (2000),
