AZ-GHS-22
Cat. No.:YN322163
产品名称: | AZ-GHS-22 |
CAS No.: | 1143020-91-0 |
Chemical Name: | 2-chloro-N-[[[6-[[3-(4-methyl-1-piperazinyl)propyl]sulfonyl]-2-benzothiazolyl]amino]carbonyl]-5-(4-morpholinyl)-benzamide |
Synonyms: | |
分子量: | 621.17306 |
分子式: | C27H33ClN6O5S2 |
SMILES: | O=C(NC1=NC2=C(S1)C=C(S(=O)(CCCN3CCN(CC3)C)=O)C=C2)NC(C4=CC(N5CCOCC5)=CC=C4Cl)=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | AZ-GHS-22 是一种有效的非 CNS 渗透性GHS-R1a反向激动剂 (IC50=0.77 nM)。 |
IC50和靶点: | |
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Solvent & Solubility: |
McCoull, W., Barton, P., Brown, A.J.H., et al.Identification, optimization, and pharmacology of acylurea GHS-R1a inverse agonistsJ. Med. Chem.57(14),6128-6140(2014)