PD 135158
Cat. No.:YN322223
产品名称: | PD 135158 |
CAS No.: | 130325-35-8 |
Chemical Name: | |
Synonyms: | CAM 1028 |
分子量: | 811.96 |
分子式: | C42H61N5O11 |
SMILES: | O[C@H]([C@H]([C@@H]([C@@H](CO)O)O)O)C[NH2+]C.O=C([O-])CCC(N[C@@H](C1=CC=CC=C1)CNC([C@](NC(O[C@@H]2C(C3(C)C)(C)CCC3C2)=O)(C)CC4=CNC5=C4C=CC=C5)=O)=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | PD 135158 (CAM 1028) 是一种选择性CCKB受体拮抗剂,对小鼠皮质 CCKB的IC50为 2.8 nM。PD 135158 表现出抗焦虑活性。 |
IC50和靶点: | [{name:"CCKBR:2.8 nM (IC50)"},{name: "CCKAR:1232 nM (IC50)"}] |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |