I-SAP
Cat. No.：YN322232
| 产品名称: | I-SAP |
| CAS No.: | 133538-58-6 |
| Chemical Name: | (5Z)-7-[(1S,2S,3S,5R)-3-[[(4-iodophenyl)sulfonyl]amino]-6,6-dimethylbicyclo[3.1.1]hept-2-yl]-5-heptenoic acid |
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| 分子量: | 531.4 |
| 分子式: | C22H30INO4S |
| SMILES: | CC1(C)[C@@H]2[C@H](C/C=C\CCCC(O)=O)[C@@H](N([H])S(C3=CC=C(I)C=C3)(=O)=O)C[C@H]1C2 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | I-SAP 是一种放射性TXA2/PGH2受体拮抗剂。I-SAP 与受体的结合被组氨酸修饰试剂二乙基焦碳酸酯 (DEPC) 抑制。 |
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Naka, M., Mais, D.E., Morinelli, T.A., et al.7-[(1R,2S,3S,5R)-6,6-Dimethyl-3-(4-iodobenzenesulfonylamino)bicyclo[3.1.1]hept-2-yl]-5(Z)-heptenoic acid: A novel high-affinity radiolabeled antagonist for platelet thromboxane A2/prostaglandin H2 receptorsJ. Pharmacol. Exp. Ther.262,632-637(1992)
