Valiglurax
Cat. No.:YN322373
| 产品名称: | Valiglurax |
| CAS No.: | 1976050-09-5 |
| Chemical Name: | |
| Synonyms: | VU0652957; VU2957 |
| 分子量: | 329.286 |
| 分子式: | C16H10F3N5 |
| SMILES: | FC(F)(F)C1=NC=CC2=C1C=CC(NC3=NNC4=C3C=CC=N4)=C2 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Valiglurax (VU0652957) 是一种口服有效的选择性mGlu4正变构调节剂,对 hmGlu4和 rmGlu4GIRK 的EC50值分别为 64.6 nM 和 197 nM。Valiglurax 是一种中枢神经系统 (CNS) 渗透剂。Valiglurax 可用于帕金森病的研究。 |
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