N-Arachidonyldopamine
Cat. No.：YN322378
CAS No. ：199875-69-9
规格
价格(RMB)
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| 产品名称: | N-Arachidonyldopamine |
| CAS No.: | 199875-69-9 |
| Chemical Name: | N-[2-(3,4-dihydroxyphenyl)ethyl]-5Z,8Z,11Z,14Z-eicosatetraenamide |
| Synonyms: | |
| 分子量: | 439.6 |
| 分子式: | C28H41NO3 |
| SMILES: | CCCCC/C=C\C/C=C\C/C=C\C/C=C\CCCC(=O)NCCc1ccc(O)c(O)c1 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | N-Arachidonyldopamine 是一种强效的、选择性的内源性CB1受体激动剂，其Ki为 250 nM。N-Arachidonyldopamine 也是一种有效的选择性TRPV1激动剂，其EC50为~50 nM。 |
| IC50和靶点: | [{name:"CB1:250 nM (Ki)"},{name: "TRPV1:~50 nM (EC50)"}] |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
Bisogno, T., Melck, D., Bobrov, M.Y., et al.N-acyl-dopamines: Novel synthetic CB1 cannabinoid-receptor ligands and inhibitors of anandamide inactivation with cannabimimetic activity in vitro and in vivoBiochem. J.351(Pt 3),817-824(2001)
