Rilmenidine phosphate
Cat. No.:YN380368
| 产品名称: | Rilmenidine phosphate |
| CAS No.: | 205437-64-5 |
| Chemical Name: | |
| Synonyms: | |
| 分子量: | 233.7 |
| 分子式: | C12H12ClN3 |
| SMILES: | C1(C2=NCCN2)=NC3=CC=CC=C3C=C1.Cl |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | BU224 hydrochloride 是一种选择性高亲和力的咪唑啉imidazoline I2受体配体,Ki为 2.1 nM。BU224 hydrochloride 有时被用作 I2受体拮抗剂。BU224 hydrochloride 具有神经保护作用,具有抗炎、抗凋亡作用。BU224 hydrochloride 可改善 5XFAD 小鼠的记忆,增大树突棘和减少 Aβ 诱导的 NMDARs 的变化。BU224 hydrochloride 可用于阿尔茨海默病研究。 |
| IC50和靶点: | |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |