RTICBM-189
Cat. No.:YN322554
| 产品名称: | RTICBM-189 |
| CAS No.: | 551909-15-0 |
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| 分子量: | 309.19 |
| 分子式: | C15H14Cl2N2O |
| SMILES: | ClC1=CC=C(NC(=O)NCCC2=CC(=CC=C2)Cl)C=C1 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | RTICBM-189 是一种有效的,可透过血脑屏障的大麻素 1 型(CB1)受体变构调节剂,在 Ca2+动员试验中pIC50为 7.54。RTICBM-189 对 hCB1和 mCB1的 pIC50分别为 5.29 和 6.25。 |
| IC50和靶点: | [{name:"CB1:7.54 (pIC50)"},{name: "hCB1:5.29 (pIC50)"},{name: "mCB1:6.25 (pIC50)"}] |
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