Orvepitant maleate
Cat. No.:YN322563
| 产品名称: | Orvepitant maleate |
| CAS No.: | 579475-24-4 |
| Chemical Name: | |
| Synonyms: | GW823296 maleate |
| 分子量: | 744.7 |
| 分子式: | C35H39F7N4O6 |
| SMILES: | 暂无 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Orvepitant maleate (GW823296 maleate) 是一种有效,选择性,口服活性且耐受性良好的neurokinin-1 (NK-1)受体拮抗剂,对人neurokinin-1受体的pKi为 10.2。Orvepitant maleate 可以穿越血脑屏障。Orvepitant maleate 可用于抑郁症和慢性顽固性咳嗽的研究。 |
| IC50和靶点: | [{name:"NK1:10.2 (pKi)"}] |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |