Iloperidone hydrochloride
Cat. No.：YN322646
CAS No. ：824393-18-2
规格
价格(RMB)
库存
| 产品名称: | Iloperidone hydrochloride |
| CAS No.: | 824393-18-2 |
| Chemical Name: | |
| Synonyms: | 阿戈美拉汀 L(+ |
| 分子量: | 393.3878 |
| 分子式: | C19H23NO8 |
| SMILES: | CC(NCCC1C2=C(C=CC(OC)=C2)C=CC=1)=O.OC([C@@H]([C@H](C(=O)O)O)O)=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Agomelatine L(+)-Tartaric acid (S-20098 L(+)-Tartaric acid) 是一种MT1和MT2受体的特异性激动剂，对 CHO-hMT1，HEK-hMT1，CHO-hMT2，HEK-hMT2 的Ki分别为 0.1，0.06，0.12 和 0.27 nM。Agomelatine L(+)-Tartaric acid 还是一种选择性的5-HT2C受体拮抗剂，在天然 (猪) 和克隆的人 5-HT2C 受体中pKi分别为 6.4 和 6.2。 |
| IC50和靶点: | [{name:"5-HT2C Receptor:6.4 (pKi, native porcine)"},{name: "5-HT2C Receptor:6.2 (pKi, human)"},{name: "hMT1:0.1 nM (Ki, CHO Cells)"},{name: "hMT1:0.06 nM (Ki, HEK Cells)"},{name: "hMT2:0.12 nM (Ki, CHO Cells)"},{name: "hMT2:0.27 nM (Ki, HEK Cells)"}] |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
