S-777469
Cat. No.:YN322802
| 产品名称: | S-777469 | 
| CAS No.: | 885496-53-7 | 
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| 分子量: | 414.47 | 
| 分子式: | C23H27FN4O2 | 
| SMILES: | 暂无 | 
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. | 
| 运输: | Room temperature in continental US; may vary elsewhere. | 
| 产品描述: | S-777469 是一种选择性,具有口服活性的大麻素 2 型受体(CB2)激动剂,Ki为 36 nM。S-777469 以剂量依赖性方式显著抑制化合物 48/80 诱导的小鼠抓挠行为。S-777469 通过CB2兴奋抑制瘙痒信号的传递,从而产生止痒作用。 | 
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