SGC-AAK1-1
Cat. No.:YN380535
CAS No. :2247894-32-0
产品名称: | SGC-AAK1-1 |
CAS No.: | 2247894-32-0 |
Chemical Name: | |
Synonyms: | SGCAAK11; SGC AAK1 1; SGC-AAK1-1; SGCAAK1-1; SGC-AAK11 |
分子量: | 427.52 |
分子式: | C21H25N5O3S |
SMILES: | O=C(C1CC1)NC2=NNC3=C2C=CC(C4=CC=CC(NS(=O)(N(CC)CC)=O)=C4)=C3 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | SGC-AAK1-1 是一种有效且选择性的AAK1(AP2 相关的激酶 1) 抑制剂,IC50为 270 nM,Ki值为 9 nM。SGC-AAK1-1 也有效抑制 BMP2K。SGC-AAK1-1 用于研究与AAK1相关的Wnt途径。 |
IC50和靶点: | |
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In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |