MAO-B-IN-9
Cat. No.:YN380543
产品名称: | MAO-B-IN-9 |
CAS No.: | 2416910-88-6 |
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分子量: | 300.4 |
分子式: | C18H24N2O2 |
SMILES: | 暂无 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | MAO-B-IN-9 (compound 16) 是一种有效的、选择性的、透过血脑屏障的、不可逆的、时间依赖性的MAO-B(单胺氧化酶 B) 抑制剂,其IC50值为 0.18 μM。MAO-B-IN-9 可防止 Aβ1-42诱导的神经元细胞死亡。MAO-B-IN-9 具有神经保护作用,其机制可能与 Aβ1-42抗聚集作用有关。 |
IC50和靶点: | [{name:"MAO-B:0.178 ± 0. μM (IC50)"}] |
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