Hemicholinium 3
Cat. No.:YN380552
| 产品名称: | Hemicholinium 3 |
| CAS No.: | 312-45-8 |
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| Synonyms: | Hemicholinium dibromide |
| 分子量: | 574.354 |
| 分子式: | C24H34Br2N2O4 |
| SMILES: | 暂无 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Hemicholinium 3 是一种竞争性的高亲和力胆碱转运蛋白 (HACU) 抑制剂,Ki值为 25 nM。Hemicholinium 3抑制乙酰胆碱 (ACh)的合成和释放,用作一种神经肌肉阻滞剂。Hemicholinium 3 抑制Epibatidine诱发的收缩和 [3H] 乙酰胆碱释放,IC50分别为 897 nM 和 693 nM。 |
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