Dienogest
Cat. No.：YN481775
CAS No. ：65928-58-7
规格
价格(RMB)
库存
| 产品名称: | Dienogest |
| CAS No.: | 65928-58-7 |
| Chemical Name: | (17α)-17-hydroxy-3-oxo-19-norpregna-4,9-diene-21-nitrile |
| Synonyms: | 地诺孕素; STS 557 |
| 分子量: | 311.42 |
| 分子式: | C₂₀H₂₅NO₂ |
| SMILES: | C[C@@]12[C@](O)(CC#N)CC[C@@]1([H])[C@]3([H])CCC4=CC(CCC4=C3CC2)=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Dienogest(STS-557)是孕酮受体激动剂，有口服的子宫内膜活性，可作用于子宫内膜异位。 |
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Sasagawa, S., Shimizu, Y., Kami, H., et al.Dienogest is a selective progesterone receptor agonist in transactivation analysis with potent oral endometrial activity due to its efficient pharmacokinetic profileSteroids73(2),222-231(2008)
Katsuki, Y., Takano, Y., Futamura, Y., et al.Effects of dienogest, a synthetic steroid, on experimental endometriosis in ratsEur. J. Endocrinol.138(2),216-226(1998)
Katsuki, Y., Shibutani, Y., Aoki, D., et al.Dienogest, a novel synthetic steroid, overcomes hormone-dependent cancer in a different manner than progestinsCancer79(1),169-176(1997)
