RIPK3-IN-1
Cat. No.:YN270830
| 产品名称: | RIPK3-IN-1 |
| CAS No.: | 2361139-70-8 |
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| 分子量: | 512.53 |
| 分子式: | C29H25FN4O4 |
| SMILES: | O=C(C1=CC=CN(C2=CC=C(F)C=C2)C1=O)NC3=CC=C(OC4=CC(NC(C5CC5)=O)=NC=C4)C(C)=C3C |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | RIPK3-IN-1 是 II 型RIPK3DFG-out 位点抑制剂,IC50为 9.1 nM。RIPK3-IN-1 抑制RIPK1和RIPK2,IC50为 5.5 和 >10 μM。RIPK3-IN-1 还是 c-Met 激酶抑制剂,IC50为 1.1 μM。 |
| IC50和靶点: | [{name:"RIPK3:9.1 nM (IC50)"}] |
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