LSN 3213128
Cat. No.:YN290079
CAS No. :1941211-99-9
产品名称: | LSN 3213128 |
CAS No.: | 1941211-99-9 |
Chemical Name: | |
Synonyms: | LSN3213128 |
分子量: | 409.46 |
分子式: | C₁₇H₁₆FN₃O₄S₂ |
SMILES: | O=C1NC=CC2=C1C=C(NS(=O)(C3=CC=C(N4CC[C@@H](O)C4)S3)=O)C(F)=C2 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | LSN 3213128 是一种选择性、非经典、口服有效的抗叶酸剂,能够有效特异性抑制氨基咪唑-4-甲酰胺核糖核苷酸甲酰转移酶 (AICARFT) 的活性,IC50值为 16 nM,在细胞中对其IC50值为 19 nM。 |
IC50和靶点: | |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |