LCH-7749944
Cat. No.:YN270180
产品名称: | LCH-7749944 |
CAS No.: | 796888-12-5 |
Chemical Name: | |
Synonyms: | GNF-PF-2356 |
分子量: | 350.41 |
分子式: | C₂₀H₂₂N₄O₂ |
SMILES: | COC1=CC(NC2=NC(NCC3OCCC3)=C4C=CC=CC4=N2)=CC=C1 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | LCH-7749944 (GNF-PF-2356) 是一种有效的PAK4抑制剂,IC50为 14.93 μM。LCH-7749944通过下调 PAK4/c-Src/EGFR/cyclin D1 途径有效抑制人胃癌细胞的增殖,并诱导凋亡 (apoptosis)。 |
IC50和靶点: | [{name:"PAK4:14.93 μM (IC50)"}] |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |