LY3295668
Cat. No.:YN290142
| 产品名称: | LY3295668 |
| CAS No.: | 1919888-06-4 |
| Chemical Name: | |
| Synonyms: | AK-01 |
| 分子量: | 489.95 |
| 分子式: | C₂₄H₂₆ClF₂N₅O₂ |
| SMILES: | O=C([C@@]1(CC2=NC(NC3=NNC(C)=C3)=CC=C2F)C[C@@H](C)N(CC4=CC=CC(Cl)=C4F)CC1)O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | LY3295668 (AK-01) 是高度特异性的Aurora-A kinase的抑制剂,其对 AurA 和 AurB 的Ki值分别为 0.8 nM 和 1038 nM。 |
| IC50和靶点: | [{name:"Aurora A:0.8 nM (IC50)"}] |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |