AKI603
Cat. No.:YN290630
| 产品名称: | AKI603 |
| CAS No.: | 1432515-73-5 |
| Chemical Name: | |
| Synonyms: | AKI603;AKI-603;AKI 603 |
| 分子量: | 409.45 |
| 分子式: | C19H23N9O2 |
| SMILES: | CN1CCN(CC1)C2=NC(=NC(=C2)NC3=N[NH]C(=C3)C)NC4=CC=C(C=C4)[N;v5](=O)=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | AKI603 是一种极光激酶 A (AurA) 抑制剂,其IC50值为 12.3 nM,被开发用于克服白血病中 BCR-ABL-T315I 耐药性突变。AKI603 对白血病细胞具有很强的抗增殖活性。 |
| IC50和靶点: | [{name:"Aurora A:12.3 nM (IC50)"}] |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |