GSK3368715
Cat. No.:YN310432
产品名称: | GSK3368715 |
CAS No.: | 1629013-22-4 |
Chemical Name: | |
Synonyms: | EPZ019997 |
分子量: | 366.54 |
分子式: | C20H38N4O2 |
SMILES: | 暂无 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | GSK3368715 (EPZ019997) 是具有口服活性的,可逆的,SAM 非竞争性 I 型蛋白精氨酸甲基转移酶(PRMTs)抑制剂 (IC50=3.1 nM (PRMT1), 48 nM (PRMT3), 1148 nM (PRMT4), 5.7 nM (PRMT6), 1.7 nM (PRMT8))。GSK3368715 (EPZ019997) 导致精氨酸甲基化状态的转变,改变了外显子的使用,具有很强的抗癌活性。 |
IC50和靶点: | |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |