HWL-088
Cat. No.:YN290716
| 产品名称: | HWL-088 |
| CAS No.: | 2378617-96-8 |
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| 分子量: | 366.38 |
| 分子式: | C22H19FO4 |
| SMILES: | CC1=CC=CC=C1C2=CC(COC3=CC=C(OCC(O)=O)C(F)=C3)=CC=C2 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | HWL-088 是一种高效的,具有口服活性的游离脂肪酸受体 1 (FFA1/GPR40) 激动剂 (EC50为 18.9 nM),并具有中等PPARδ活性 (EC50为 570.9 nM)。HWL-088 改善葡萄糖和脂质代谢,并具有抗糖尿病作用。 |
| IC50和靶点: | [{name:"PPARδ:570.9 nM (EC50)"},{name: "FFAR1/GPR40:18.9 nM (EC50)"}] |
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