PF-07220060
Cat. No.:YN290717
| 产品名称: | PF-07220060 |
| CAS No.: | 2380321-51-5 |
| Chemical Name: | |
| Synonyms: | CDK4/6-IN-6 |
| 分子量: | 463.93 |
| 分子式: | C22H27ClFN5O3 |
| SMILES: | 暂无 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | PF-07220060 (CDK4/6-IN-6; example A94) 是一种有效的CDK4/CDK6抑制剂,对CDK4/Cyclin D1 和 CDK6/Cyclin D3 的 Ki 值为 0.6 nM 和 13.9 nM。 |
| IC50和靶点: | [{name:"Cdk4/cyclin D1:0.6 nM (Ki)"},{name: "cdk6/cyclin D3:13.9 nM (Ki)"}] |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |