Bobcat339 hydrochloride
Cat. No.:YN310556
| 产品名称: | Bobcat339 hydrochloride |
| CAS No.: | 2436747-44-1 |
| Chemical Name: | |
| Synonyms: | Bobcat339 HCl |
| 分子量: | 334.2 |
| 分子式: | C16H13Cl2N3O |
| SMILES: | C1=CC=C(C=C1)C2=CC(=CC=C2)N3C=C(C(=NC3=O)N)Cl |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Bobcat339 hydrochloride 是一种有效的、选择性的基于胞嘧啶的TET酶抑制剂,抑制TET1和TET2的IC50值分别为 33 μM 和 73 μM。Bobcat339 hydrochloride 可用于表观遗传学领域研究,并且可作为靶向 DNA 甲基化和基因转录新疗法的起点。 |
| IC50和靶点: | [{name:"TET1:33 μM (IC50)"},{name: "TET2:73 μM (IC50)"}] |
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| Clinical Trial: | |
| Solvent & Solubility: |